Design and synthesis of some furan derivatives and Its lsosteres of anticipated antitumor activity / Shaimaa Mohamed Abdelrahman ; Supervised Samir M. Elmoghazy , Nahed M. Eid , Sahar M. AbouSeri
Material type:
- تصميم و تشييد بعض مشتقات الفيوران و متشابهاتها من المتوقع أن يكون لها فاعلية ضد الأورام [Added title page title]
- Issued also as CD
Item type | Current library | Home library | Call number | Copy number | Status | Barcode | |
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قاعة الرسائل الجامعية - الدور الاول | المكتبة المركزبة الجديدة - جامعة القاهرة | Cai01.08.05.Ph.D.2014.Sh.D (Browse shelf(Opens below)) | Not for loan | 01010110066185000 | ||
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مخـــزن الرســائل الجـــامعية - البدروم | المكتبة المركزبة الجديدة - جامعة القاهرة | Cai01.08.05.Ph.D.2014.Sh.D (Browse shelf(Opens below)) | 66185.CD | Not for loan | 01020110066185000 |
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Thesis (Ph.D.) - Cairo University - Faculty of Pharmacy - Department of Pharmaceutical Chemistry
In this thesis, novel series of colchicine binding site inhibitors (CBSIs) were designed. Molecular modeling techniques were used to support the design. Chalcones derivatives IIa - d, cyclohexenone derivatives IIIa,b, IVa,b, cyanopyridine derivatives VIa, b, isoxazoline derivatives VIIa - d, pyrazoline derivatives VIIIa, b, IXa, b, Xa - f, XIa, b and XIIa - f were synthesized. Eight target compounds were evaluated for antitumor activity at National cancer institute, NCI, maryland, USA against several cell lines. Twenty four target compounds were evaluated for antitumor activity and their ability to inhibit tubulin polymerization against leukemia SR cell line at Vacsera, Egypt
Issued also as CD
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