Design of novel diarylheterocycles with potential phosphodiesterase inhibitory and anticancer properties / Mahmoud Amr Mahmoud Elnaggar ; Supervised Ashraf H. Abadi
Material type: TextLanguage: English Publication details: Cairo : Mahmoud Amr Mahmoud Elnaggar , 2011Description: 88Leaves : charts , facsimiles ; 30cmOther title:- تصميم مركبات داى أريل جديدة غير متجانسة الحلقة مثبطة لإنزيم الفوسفوداى إستريز وذات خواص مضادة للسرطان [Added title page title]
Item type | Current library | Home library | Call number | Status | Date due | Barcode | |
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Thesis | قاعة الثقاقات الاجنبية - الدور الثالث | المكتبة المركزبة الجديدة - جامعة القاهرة | Cai01.34.M.Sc.2011.Ma.D (Browse shelf(Opens below)) | Not for loan | 01010110060230000 |
Thesis (M.Sc.) - German University - Faculty of Postgraduate Studies and Scientific Research - Department of Pharmaceutical Chemistry
Many Cyanopyridines and Cyanopyiridones were reported to have cardiotonic and anticancer properties . The first activity is mediated through the inhibition of PDEIII leading to elevation of secondary messengers namely cAMP and cGMP , the latter activity were shown to be due to the inhibitory action on targets that are over - expressed in cancerous cells such as PIM1 Kinase and the anti - apoptotic protein ; Survivin leading to growth inhibition of cancer cells
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