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040 _aEG-GICUC
_beng
_cEG-GICUC
_dEG-GICUC
_erda
041 0 _aeng
_beng
_bara
049 _aDeposit
082 0 4 _a546
092 _a546
_221
097 _aM.Sc
099 _aCai01.12.09.M.Sc.2024.Ya.D
100 0 _aYasser Abo Elfotoh Elsayed,
_epreparation.
245 1 0 _aDesign, structual inspection, pharmaceutical and interaction with DNA studies of some transition metal chelates derived from ciprofloxacin /
_cby Yasser Abo Elfotoh Elsayed ; Supervisors Prof.Dr.Gehad Genidy Mohamed, Prof.Dr.Ahmed Mohammed Abu-Dief.
246 1 5 _aتصميم وفحص الشكل التركيبي ودراسات صيدلانية والتداخل مع الحمض النووي الديؤكسي ريبوزي لبعض مخلبيات العناصر الانتقاليه والمشتقه من السيبروفلوكساسين
264 0 _c2024.
300 _a164 pages :
_billustrations ;
_c25 cm. +
_eCD.
336 _atext
_2rda content
337 _aUnmediated
_2rdamedia
338 _avolume
_2rdacarrier
502 _aThesis (M.Sc)-Cairo University, 2024.
504 _aBibliography: pages 144-163.
520 3 _aNovel compounds with pharmacological activity were synthesized from Pd [II], Fe [III], Cr [II], Ni [II] and Cu [II] ions with 1_Cyclopropyl _ 6- fluoro_ 4_ (2-hydroxy-phenylimino)_7_ piperazin _1_yl_1,4_dihydro_quinoline_ 3_ carboxylic acid (CFAP). The ligand's NH and OH groups allowed it to interact with the metals as a neutral tri-dentate. The novel compounds were described using (1H and 13C NMR spectra),( FT- IR spectrums), (TGA), ultraviolet _ visible light), (conductance of molecules), and CHN-analysis. Additionally, the pH profile of the CFAP complexes indicated great stability, and the complexes' stability constant was discovered in the solution. To extract important properties for CFAP and its complexes, computational research was used CFAPCu , CFAPCr, CFAPNi, and CFAPFe have octahedral geometry, while CFAPPd has square planar geometry. To investigate the molecular geometry, density functional theory calculations (DFT) were carried out. The molar ratio and continuous fluctuation data confirmed that the (M:L) ratio was (1:1). In vitro tests were conducted to evaluate schiff base's antimicrobial action ligand and its metal chelates against fungal and bacterial infections. The findings showed that the antimicrobial efficacy is as follows: when CFAPPd is compared to Fluconazol and Ofloxacin as reference medications, it is the highly inhibitor complex. The novel The ligands and their complexes in vitro carcinogenic potential in opposition to the [ Hep_G2 , MCF_7 , and HCT_116 ] cell lines was also studied. As compared to the medication vinblastine, the results once again demonstrated that CFAPPd is the most active agent. Moreover, the complexes demonstrated strong reactivity in capturing free radicals when their antioxidant activity was investigated. Viscosity, spectral investigations, and gel electrophoreses were used to identify the interaction between metal chelates and DNA. Every examined compound is shown to be an enthusiastic DNA binder by viscosity and spectrophotometric titration investigations. The heightened hydrophobic and electrostatic interactions between aromatic rings could be the cause of this. Ultimately, these compounds could be regarded as promising bioactive substances. Novel compounds with pharmacological activity were synthesized from Pd(II), Fe(III), Cr(III), Ni(II) and Cu(II) ions with 4-[2-(3-Carboxy-1- cyclopropyl-6-fluoro-7-piperazin-1-yl-2,3-dihydro-1H-quinolin-4- ylideneamino)-phenylimino]-1-cyclopropyl-6-fluoro-7-piperazin-1-yl-1,4- dihydro-quinoline-3-carboxylic acid (CFPD). The newly synthesized compounds have been investigated by 1H- and 13C-NMR spectra, FT-IR spectra, CHN analyses, TG, UV-Vis, and molar conductivity. In addition, the pH-profile of the CFPD complexes showed remarkable stability, and a stability constant was identified in solution. To extract significant characteristics for CFPD and its complexes and to investigate the molecular geometry, computational analysis occurred. Through its NH and OH groups, the ligand interacted with the metal ions as a neutral bidentate that formed CFPD-Pd(II) complex has square planar geometry, CFPD-Cu(II), CFPD- Cr(III), CFPD-Ni(II) and CFPD-Fe(III) complexes have octahedral geometry. The (M:L) ratio of 1:1 was shown by the results of the molar ratio and continuous variation procedures. A variety of fungi and viral pathogens were used to investigate the in vitro antibacterial activity of the Schiff base ligand and its complexes with metals. The results revealed that the antimicrobial efficacy followed the order: CFPD-Pd(II) complex is the highly inhibitor complex compared to fluconazol and ofloxacin as reference drugs. The in-vitro cytotoxic activity of the new ligand and its complexes was also investigated against Hep-G2, MCF-7 and HCT-116 cell lines. The results showed again that CFPD-Pd(II) complex is the highest active agent compared to vinblastine drug. In addition, the complexes showed high reactivity in catching free radicals when their antioxidant activity was examined. By the application of viscosity, spectrum analysis, and gel electrophoreses, the interaction among metal chelates and DNA was determined. Studies on viscosity and spectrophotometric titration showed that every substance in test is a strong DNA binder. Increased hydrophobic and electrostatic interactions between aromatic rings could be the cause of this. In conclusion, these complexes have the potential to be effective bioactive agents.
520 3 _aتعتبر مركبات الفلوروكينولين من المركبات الكيميائية الهامة والتى تلعب دوراً مميزاً فى مجال الكيمياء التناسقية وذلك لقدرتها على تكوين متراكبات مستقرة بسهولة مع كثير من أيونات العناصر الإنتقالية بالإضافة إلى ذلك ترجع أهميتها لكونها تستخدم كمضادات للبكتريا والفطريات، كما أنها لها قدرة فائقة علي الارتباط مع الحمض النووي الديؤكسي ريبوزي مما يؤهلها لأن تستخدم كمضادات قوية للفيروسات والأورام السرطانية وكذلك لقدرتها على إقتناص أيونات المعادن مما يجعل لها دورا هاما فى الكيمياء التحليلية والصناعية حيث أنها تستخدم فى تنقية مياه الشرب وتخليصها من أيونات المعادن الثقيلة وكذلك تستخدم لمقاومة تاكل المعادن مثل الحديد. واجتذب سيبروفلوكساسين أيضًا اهتمامًا من المجتمع العلمي بسبب نشاطه في موت الخلايا المبرمج ومضاد التكاثر في العديد من خطوط السرطان. وبناءا على ما سبق ذكره فإن الأهداف الرئيسية من هذه الرسالة جاءت علي النحو التالي: • تحضير بعض ليجيندات الإيمين المحتوية على السيبروفلوكساسين ثلاثية ورباعية العطاء • تحضير المتراكبات مع بعض أيونات العناصر الإنتقالية ثنائية التكافؤ مثل Pd(II), Ni(II) and Cu(II) وثلاثية التكافؤ مثل Fe(III), Cr(III), والتى ثبت ان لها فاعلية بيولوجية ضد العديد من الخلايا البكتيرية والفطريات والخلايا السرطانية والشقوق الحرة.
530 _aIssues also as CD.
546 _aText in English and abstract in Arabic & English.
650 0 _aInorganic
653 1 _aSchiff base complexes
_aThermal analyses (TG and DTG)
_aDFT
_aantibacterial activity
_aantioxidant activity
_aMolecular docking studies.
700 0 _aGehad Genidy Mohamed
_ethesis advisor.
700 0 _aAhmed Mohammed Abu-Dief
_ethesis advisor.
900 _b01-01-2024
_cGehad Genidy Mohamed
_cAhmed Mohammed Abu-Dief
_UCairo University
_FFaculty of Science
_DDepartment of Chemistry
905 _aShimaa
_eEman Ghareb
942 _2ddc
_cTH
_e21
_n0
999 _c173593