000 01894nam a2200361 a 4500
003 EG-GiCUC
005 20250223025912.0
008 090720s2009 ua h f m 000 0 eng d
040 _aEG-GiCUC
_beng
_cEG-GiCUC
041 0 _aeng
049 _aDeposite
097 _aPh.D
099 _aCai01.08.04.Ph.D.2009.Ha.C
100 0 _aHala Bakr Ali Elnassan
245 1 0 _aComputer-based drug design and synthesis of certain pyrazolopyrimidine and bis(pyrimidinyI) methane derivatives as potential antineoplastic agents /
_cHala Bakr Ali Elnassan ; Supervised Mervat Mostafa Elenany , Mona Monir Kamel , Omneya Mahmoud Khalil
246 1 5 _aتصميم وتشييد بعض مشتقات من البيرازولوبيريميدين وثنائى بيريميدنيل ميثان كمضادات للاورام السرطانية
260 _aCairo :
_bHala Bakr Ali Elnassan ,
_c2009
300 _a132P. :
_bfacsimiles ;
_c25cm
502 _aThesis (Ph.D.) - Cairo University - Faculty of Pharmacy - Department of Organic chemistry
520 _aThe study comprises a survey on the cyclin dependent kinases(CDKs) and their inhibtors.The thesis involves the design docking study and synthesis of some pyrazolo[3,4-d] pyrimidin-4-one,pyrazolo[1,5-a] pyrimidine and bis(6-aminopyrimidin-5-y1) (substituted pheny1) methane derivatives as CDK2 inhibitors to be investigated as new antineoplastic agents
530 _aIssued also as CD
653 4 _aAntineoplastic activity
653 4 _aBis(6-aminopyrimidin-5-y1) (substituted pheny1) methane
653 4 _aPyrazolo[3,4-d] pyrimidin-4-one
700 0 _aMervat Mostafa Elenany ,
_eSupervisor
700 0 _aMona Monir Kamel ,
_eSupervisor
700 0 _aOmneya Mahmoud Khalil ,
_eSupervisor
856 _uhttp://172.23.153.220/th.pdf
902 _a1
905 _aFatma
_eCataloger
905 _aNazla
_eRevisor
942 _2ddc
_cTH
999 _c23175
_d23175