000 02474cam a2200349 a 4500
003 EG-GiCUC
005 20250223031537.0
008 160814s2016 ua dh f m 000 0 eng d
040 _aEG-GiCUC
_beng
_cEG-GiCUC
041 0 _aeng
049 _aDeposite
097 _aPh.D
099 _aCai01.08.04.Ph.D.2016.Mo.A
100 0 _aMohamed Tawfik Mohamed Nemr
245 1 0 _aApplication of solid phase technique in the synthesis of certain heterocycles of expected pharmaceutical interest /
_cMohamed Tawfik Mohamed Nemr ; Supervised Mohamed Mohsen Ismail , Hanan Mohamed Refaat , Mona Monir Kamel
246 1 5 _aتطبيق تقنية الطور الجامد في تشييد مركبات معينة غير متجانسة الحلقة من المتوقع أن يكون لها أهمية
260 _aCairo :
_bMohamed Tawfik Mohamed Nemr ,
_c2016
300 _a185 P. :
_bcharts , facsimiles ;
_c25cm
502 _aThesis (Ph.D.) - Cairo University - Faculty of Pharmacy - Department of Organic Chemistry
520 _aThis thesis comprises four chapters. The first chapter is an introduction which includes the solid phase synthesis and biological activity of benzimidazoles, quinoxalines and isoalloxazines. The second chapter clarifies the objectives of the work and schemes designed for the preparation of the target compounds. The third chapter deals with the theoretical discussion of the experimental work, molecular docking and results of cytotoxic activity. The fourth chapter includes the experimental part of the thesis which contains the detailed procedures used for the synthesis of the target compounds and intermediates, in addition to their physical properties, their elemental analyses and spectral data. Moreover, it includes the docking steps of all compounds. The in vitro cytotoxic activity of the synthesized compounds on breast cancer cell line (MCF-7), human hepatic cell line (HEPG2) and human colorectal cell line (HCT116) compared with doxorubicin as a reference anticancer agent is also included in this chapter
530 _aIssued also as CD
653 4 _aBenzimidazoles
653 4 _aQuinoxalines
653 4 _aSolid phase synthesis
700 0 _aHanan Mohamed Refaat ,
_eSupervisor
700 0 _aMohamed Mohsen Ismail ,
_eSupervisor
700 0 _aMona Monir Kamel ,
_eSupervisor
856 _uhttp://172.23.153.220/th.pdf
905 _aNazla
_eRevisor
905 _aSamah
_eCataloger
942 _2ddc
_cTH
999 _c57438
_d57438