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008 170119s2016 ua dh f m 000 0 eng d
040 _aEG-GiCUC
_beng
_cEG-GiCUC
041 0 _aeng
049 _aDeposite
097 _aPh.D
099 _aCai01.08.08.Ph.D.2016.Mu.E
100 0 _aMugahed Mohammed Ahmed Algamrah
245 1 0 _aEnhancement of solubility and bioavailability of glimepiride using nanotechnology /
_cMugahed Mohammed Ahmed Algamrah ; Supervised Ahmed Abdelbary Abderahman , Omneya Mohamed Abdelkader
246 1 5 _aتحسين الأذابة والأتاحة الحيوية لعقار الجليمبيرايد بأستخدام تكنولوجيا النانو
260 _aCairo :
_bMugahed Mohammed Ahmed Algamrah ,
_c2016
300 _a166 P. :
_bcharts , facsimiles ;
_c25cm
502 _aThesis (Ph.D.) - Cairo University - Faculty of Pharmacy - Department of Pharmaceutics
520 _aMany of Poorly aqueous soluble drugs including antihypertensive agents, antidiabetic agents and anti cancer agents require novel delivery technologies that will enhance their GIT absorption, maximize their bioavailability and lead to efficient therapeutic effect. Over the past two decades, there has been a steady rise in the number of commercially available nanoparticle (NP), solid nanodispersion and solid lipid nanoparticles (SLNs) therapeutics as novel delivery technologies intended to enhance the GIT absorption, maximize the bioavailability and lead to efficient therapeutic effect of poorly aqueous soluble drugs. Glimepiride is considered as new generation of sulfonyl urea and administered orally. Its main draw back is its poor solubility. Glimepiride, chemically described as 1-[[4-[2-(3-ethyl-4-methyl-2-oxo-3-pyrroline-1- carboxamide) ethyl] phenyl] sulphonyl] -3-(trans-4-methylcyclohexyil) urea, is water insoluble oral antidiabetic drug from the sulfonylurea class, which is widely used in the treatment of type 2 diabetes. Glimepiride was selected as drug candidate, as it is not available in such dosage forms and thus, to enhance safety and efficacy of Glimepiride, achieve better compliance, solve the problem of solubility, absorption and bioavailability. To achieve these goals, the work in our thesis is divided into four chapters
530 _aIssued also as CD
653 4 _aEnhancement of solubility and bioavailability
653 4 _aGlimepiride
653 4 _aNanotechnology
700 0 _aAhmed Abdelbary Abdelrahman ,
_eSupervisor
700 0 _aOmneya Mohamed Abdelkader ,
_eSupervisor
856 _uhttp://172.23.153.220/th.pdf
905 _aEnas
_eCataloger
905 _aNazla
_eRevisor
942 _2ddc
_cTH
999 _c57770
_d57770