000 02486cam a2200349 a 4500
003 EG-GiCUC
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008 170823s2016 ua dho f m 000 0 eng d
040 _aEG-GiCUC
_beng
_cEG-GiCUC
041 0 _aeng
049 _aDeposite
097 _aPh.D
099 _aCai01.08.04.Ph.D.2016.So.S
100 0 _aSoha Hussein Emam Mabrouk
245 1 0 _aSynthesis and evaluation of certain diaryl substituted heterocyclic compounds as potential anticancer agents /
_cSoha Hussein Emam Mabrouk ; Supervised Salwa Elsayed Mohamed Elmeligie , Nadia Abdalla Khalil , Eman Mohamed Ahmed
246 1 5 _aتشييد و تقييم بعض المركبات الحلقية الغير متجاًنسة المستبدلة بثنائى الآريل ذات تاثير محتمل كمضادات للسرطان
260 _aCairo :
_bSoha Hussein Emam Mabrouk ,
_c2016
300 _a06 P. :
_bcharts , facsimiles , photographs ;
_c25cm
502 _aThesis (Ph.D.) - Cairo University - Faculty of Pharmacy - Department of Organic Chemistry
520 _aThis thesis comprises five chapters. The first one is an introduction which includes a brief literature survey on the synthesis, anticancer and antimitotic activities of 2-pyrazolines, 1,3,4-oxadiazoles and pyridines. The second chapter clarifies the aim of the work and the schemes adopted for the preparation of the target compounds. The third chapter deals with the theoretical discussion of the experimental work. The fourth chapter consists of the experimental part of the thesis which contains detailed procedures used for the synthesis of the target compounds, as well as the physical properties and detailed data obtained from elemental and spectral analyses. The fifth chapter includes discussion of the anticancer results compared to standard antimitotic agent colchicine, as well as a brief account on the results of the docking study and the correlation between these results and anticancer activity. It also includes the procedures of anticancer testing as well as the docking steps followed
530 _aIssued also as CD
653 4 _a1, 3, 4-oxadiazole
653 4 _a2-pyrazoline
653 4 _aPyridine
700 0 _aEman Mohamed Ahmed ,
_eSupervisor
700 0 _aNadia Abdalla Khalil ,
_eSupervisor
700 0 _aSalwa Elsayed Mohamed Elmeligie ,
_eSupervisor
856 _uhttp://172.23.153.220/th.pdf
905 _aNazla
_eRevisor
905 _aSamia
_eCataloger
942 _2ddc
_cTH
999 _c62124
_d62124