000 02455cam a2200349 a 4500
003 EG-GiCUC
005 20250223032550.0
008 200831s2020 ua d f m 000 0 eng d
040 _aEG-GiCUC
_beng
_cEG-GiCUC
041 0 _aeng
049 _aDeposite
097 _aPh.D
099 _aCai01.12.10.Ph.D.2020.Am.S
100 0 _aAmna Mohamed Abdella
245 1 0 _aSynthesis and characterization of some novel bis-heterocyclic derivatives /
_cAmna Mohamed Abdella ; Supervised Ahmed Helmy Mahmoud Elwahy , Ismail Abdelshafy Abdelhamid , Amr Mohamed Abdelmoniem
246 1 5 _aتشييد و توصيف بعض المشتقات الحلقية غير المتجانسة الثنائية والمتماثلة الجديدة
260 _aCairo :
_bAmna Mohamed Abdella ,
_c2020
300 _a151 P. :
_bcharts ;
_c25cm
502 _aThesis (Ph.D.) - Cairo University - Faculty of Science - Department of Organic Chemistry
520 _aPart 1: Novel bis(1,4-dihydropyridine-3,5-dicarbonitrile) derivatives linked to arene core via ethter amide or ester-amide linkages were prepared by the reaction of the bis-aldehydes with four equivalents of 3-aminocrotononitrile in the presence of acid catalyst. The molecular docking simulation studies indicated that, the prepared compounds bind to the active site of cellular inhibitor apoptotic protein (cIAP1-BIR3).Part 2: One-pot three-component reaction of bis(aldehydes) with 6-aminouracil in boiling acetic acid afforded tetrakis(6-aminopyrimidine-2,4-diones) or bis(tetraoxodecahydropyrido [2,3-d:6,5-d']dipyrimidines) depending on the reaction conditions.Part 3: A synthesis of novel bis(1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile), bis(4Hchromene- 3-carbonitrile) and bis(dihydropyrano[3,2-c]chromene) via multicomponent reactions of the appropriate bis-aldehyde with two equivalents of both of malononitrile and 3- methylpyrazol-5-one, dimedone or 4-hydroxycoumarin in a basic solution
530 _aIssued also as CD
653 4 _aBis(1,4-dihydropyridine-3,5- dicarbonitrile)
653 4 _aBis(aldehydes) linked to amide linkages
653 4 _aTetrakis(6-aminouracil-5-yl)methanes
700 0 _aAhmed Helmy Mahmoud Elwahy ,
_eSupervisor
700 0 _aAmr Mohamed Abdelmoniem ,
_eSupervisor
700 0 _aIsmail Abdelshafy Abdelhamid ,
_eSupervisor
856 _uhttp://172.23.153.220/th.pdf
905 _aNazla
_eRevisor
905 _aShimaa
_eCataloger
942 _2ddc
_cTH
999 _c77469
_d77469