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040 _aEG-GiCUC
_beng
_cEG-GiCUC
041 0 _aeng
049 _aDeposite
097 _aM.Sc
099 _aCai01.08.03.M.Sc.2021.Mi.A
100 0 _aMina Wadie Ibrahim
245 1 0 _aAnalytical study of some drugs treating benign prostatic hyperplasia /
_cMina Wadie Ibrahim ; Supervised Ezzat Mohamed Abdelmoety , Soheir Abdelfattah Ahmed Omar , Mamdouh Reda Rezk
246 1 5 _aدراسة تحليلية لبعض الأدوية المعالجة لتضخم البروستاتا الحميد
260 _aCairo :
_bMina Wadie Ibrahim ,
_c2021
300 _a421 P. :
_bcharts ;
_c25cm
502 _aThesis (M.Sc.) - Cairo University - Faculty of Pharmacy - Department of Analytical Chemistry
520 _aThis thesis is concerned with the quantitative determination of some drugs used for treatment of benign prostatic hyperplasia and other coincident diseases. In this thesis, two binary mixtures were studied, separately, in their new pharmaceutical formulations. The first mixture contains Tamsulosin Hydrochloride (TAM) and Tadalafil (TAD), while the second one contains Alfuzosin Hydrochloride (ALF) and Solifenacin Succinate (SOL).The aim of this work was to develop different analytical methods that are characterized by simplicity, accuracy and appropriate degree of sensitivity for the analysis of the above-mentioned drugs in their pure forms, in their pharmaceutical formulations and in the presence of their degradation products and/or potential impurities. Smart UV-spectrophotometric, high-performance thin layer chromatographic (HPTLC) and high-performance liquid chromatographic (HPLC) methods were developed for the analysis of the first mixture (TAM and TAD). Moreover, the principles of green chemistry and Quality-by-Design approach were successfully implemented throughout the chromatographic separation.The greenness profile was assessed via several green metrics as GlaxoSmithKline solvent sustainability guide, environmental, health and safety (EHS) tool, national environmental methods index (NEMI) and Eco-Scale. Additionally, the stability of the two cited drugs was investigated under different stress conditions in accordance with ICH guidelines followed by developing stability-indicating high-performance thin layer chromatographic and high-performance liquid chromatographic methods.The second mixture (ALF and SOL) was assayed by eco-friendly UV-spectrophotometric and Quality-by-Design based HPLC methods in their binary mixtures. In addition, the two enantiomers of ALF were successfully separated along with SOL using 50-mm chiral column and ethanol as green organic solvent.The method was statistically optimized through experimental design. Moreover, stability-indicating high-performance thin layer chromatographic and high-performance liquid chromatographic methods were developed for the simultaneous determination of Alf and SOL along with their official impurities induced via stress stability studies
530 _aIssued also as CD
653 4 _aAlfuzosin hydrochloride
653 4 _aChromatography
653 4 _aExperimental design
700 0 _aEzzat Mohamed Abdelmoety ,
_eSupervisor
700 0 _aMamdouh Reda Rezk ,
_eSupervisor
700 0 _aSoheir Abdelfattah Ahmed Omar ,
_eSupervisor
856 _uhttp://172.23.153.220/th.pdf
905 _aNazla
_eRevisor
905 _aShimaa
_eCataloger
942 _2ddc
_cTH
999 _c80387
_d80387